2. Immunology/Inflammation
  3. COX
  4. Timegadine hydrochloride

Timegadine hydrochloride  (Synonyms: SR1368 hydrochloride)

目录号: HY-100125A
产品使用指南 技术支持

Timegadine hydrochloride (SR1368 hydrochloride) 是 Timegadine (HY-100125) 的盐酸盐形式。Timegadine hydrochloride 是口服有效的 COX 和 脂氧合酶 (lipo-oxygenase) 的抑制剂，可抑制兔血小板和大鼠脑中的 COX，IC50 分别为 5 nM 和 20 μM，可抑制马和兔血小板中的脂氧合酶，IC50 为 100 μM。Timegadine hydrochloride 具有抗关节炎活性。

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Timegadine hydrochloride Chemical Structure

Timegadine hydrochloride Chemical Structure

CAS No. : 71080-06-3

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Other Forms of Timegadine hydrochloride:

Timegadine hydrochloride 相关抗体

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COX COX-1 COX-2 COX-3

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Timegadine hydrochloride (SR1368 hydrochloride) is the hydrochloride salt form of Timegadine (HY-100125). Timegadine hydrochloride is an orally active inhibitor for COX and lipo-oxygenase, that inhibits COX in washed rabbit platelets and rat brain with IC50 of 5 nM and 20 μM, inhibits lipo-oxygenase in in horse and washed rabbit platelets with IC50 of 100 μM. Timegadine hydrochloride exhibits anti-arthritis activity[1].

分子量

401.96

Formula

C20H24ClN5S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Timegadine hydrochloride 相关分类

  • 摩尔计算器

  • 稀释计算器

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

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× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Timegadine71080-06-3SR1368SR 1368SR-1368COXCyclooxygenaseorally activeanti-arthritisInhibitorinhibitorinhibit

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目录号：
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