Endothelin Receptor Inhibitors

ET_A

ET_B

Endothelin Receptor Agonists, Antagonists & Activators

Product Name	ET_A	ET_B	Purity
Endothelin 1 (swine, human)	ET_A	ET_B	99.12%
Macitentan	ET_A	ET_B	99.95%
Ambrisentan	ET_A		99.95%
Edonentan	ET_A, Ki: 10 pM	ET_B, Ki: 810 nM
BQ-123	ET_A		99.78%
BQ-788 sodium salt		ET_B	98.56%
Sulfisoxazole	ET_A, IC₅₀: 0.60 μM	ET_B, IC₅₀: 22 μM	99.90%
Zibotentan	ET_A, Ki: 13 nM		98.19%
Aprocitentan	ET_A, IC₅₀: 3.4 nM ET_A, pA2: 6.7	ET_B, IC₅₀: 987 nM ET_B, pA2: 5.5	99.98%
A-192621	ET_A, IC₅₀: 4280 nM ET_A, Ki: 5600 nM	ET_B, IC₅₀: 4.5 nM ET_B, Ki: 8.8 nM	99.85%
Tezosentan	ET_A, pA2: 9.5	ET_B, pA2: 7.7	98.79%
IRL-1620 TFA		ET_B	99.74%
IRL 2500	ET_A, IC₅₀: 94 nM	ET_B, IC₅₀: 1.3 nM	≥99.0%
Nebentan potassium	ET_A, Ki: 0.679 nM	ET_B, Ki: 569 nM	99.53%
Ro 46-8443	ET_A, IC₅₀: 6800 nM	ET_B, IC₅₀: 34-69 nM	99.24%
Nebentan	ET_A, Ki: 0.697 nM	ET_B, Ki: 569 nM	99.67%
Macitentan-d₄	ET_A	ET_B	98.03%
IRL-1620		ET_B
BMS 182874	ET_A, IC₅₀: 0.15 μM ET_A, Ki: 0.055 μM		99.85%
ABT-546	ET_A, Ki: 0.46 nM
Ambrisentan sodium	ET_A
Aprocitentan-d₄	ET_A, IC₅₀: 3.4 nM ET_A, pA2: 6.7	ET_B, IC₅₀: 987 nM ET_B, pA2: 5.5
CI-1020	ET_A, IC₅₀: 0.3 nM
Sarafotoxin S6a	ET_A	ET_B
BMS-193884	ET_A, Ki: 1.4 nM	ET_B, Ki: 18700 nM
[Ala1,3,11,15]-Endothelin (53-63) (TFA)		ET_B
Sarafotoxin S6a TFA	ET_A	ET_B
Endothelin 1 (swine, human), Alexa Fluor 488-labeled	ET_A	ET_B
Sulfisoxazole diethanolamine	ET_A, IC₅₀: 0.60 μM	ET_B, IC₅₀: 22 μM
BQ-3020		ET_B, IC₅₀: 0.2 nM
Edonentan hydrate	ET_A, Ki: 10 pM
ATZ-1993	ET_A, pKi: 8.69	ET_B, pKi: 7.20
FR139317	ET_A
ZD-1611	ET_A

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