2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Adrenergic Receptor
  4. Etoperidone

Etoperidone 是一种抗抑郁剂，是一种具有口服活性的血清素 (serotonin) 和去甲肾上腺素 (nor-adrenaline) 再摄取拮抗剂。Etoperidone 对 5-HT2 受体、α1-肾上腺素受体 (α1-adrenergic receptor)、5-HT1A 受体和 α2-肾上腺素受体 (α2-adrenergic receptor) 的 Kd 值分别为 36 nM、38 nM、85 nM 和 570 nM。

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Etoperidone Chemical Structure

Etoperidone Chemical Structure

CAS No. : 52942-31-1

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Other Forms of Etoperidone:

Etoperidone 相关抗体

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5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

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α adrenergic receptor β adrenergic receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Etoperidone, an antidepressant agent, is an orally active serotonin and nor-adrenaline re-uptake antagonist. Etoperidone shows Kd values of 36 nM, 38 nM, 85 nM, and 570 nM for 5-HT2 receptor, α1-adrenergic receptor, 5-HT1A receptor, and α2-adrenergic receptor, respectively[1][2].

IC50 & Target[2]

5-HT1A Receptor

85 nM (Kd)

5-HT2A Receptor

36 nM (Kd)

α1-adrenergic receptor

38 nM (Kd)

α2-adrenergic receptor

570 nM (Kd)

分子量

377.91

Formula

C19H28ClN5O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Etoperidone 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Etoperidone52942-31-15-HT ReceptorAdrenergic ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorBeta Receptor5-HT2 receptor α1-adrenergic receptor5-HT1A receptor α2-adrenergic receptorantidepressant agentInhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-106617
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