1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. P2X Receptor
  4. P2X Receptor Inhibitors

P2X Receptor Inhibitors

P2X1 Receptor

P2X2 Receptor

P2X3 Receptor

P2X4 Receptor

P2X7 Receptor

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

P2X Receptor Inhibitors, Agonists, Antagonists & Activators
Product Name P2X1 Receptor P2X2 Receptor P2X3 Receptor P2X4 Receptor P2X7 Receptor Purity
BzATP triethylammonium salt
p2x1 Receptor
 
P2X3 Receptor
P2X4 Receptor
P2X7 Receptor
Sodium metatungstate        
P2X7 Receptor
A-740003        
P2X7 Receptor
99.59%
NF449 octasodium
p2x1 Receptor
        ≥99.0%
KN-62        
P2X7 Receptor
99.45%
HEI3090        
P2X7 Receptor
99.04%
Aurintricarboxylic acid
p2x1 Receptor, IC50: 8.6 nM
 
P2X3 Receptor, IC50: 72.9 nM
   
A 438079 hydrochloride        
P2X7 Receptor
99.92%
A 438079        
P2X7 Receptor
99.88%
5-BDBD      
P2X4 Receptor
  99.94%
Gefapixant    
P2X3 Receptor
    99.33%
α,β-Methylene-ATP trisodium
p2x1 Receptor
 
P2X3 Receptor
 
P2X7 Receptor
99.75%
JNJ-47965567        
P2X7 Receptor
99.79%
PPADS tetrasodium
p2x1 Receptor
       
JNJ-55308942        
P2X7 Receptor
99.92%
AZD9056 hydrochloride        
P2X7 Receptor
98.82%
BAY-1797      
P2X4 Receptor
  99.42%
AZ10606120 dihydrochloride        
P2X7 Receptor
99.38%
A-317491    
P2X3 Receptor
    98.77%
A-804598        
P2X7 Receptor
98.55%
PPNDS tetrasodium
p2x1 Receptor
       
Minodronic acid  
P2X2 Receptor
P2X3 Receptor
    99.67%
P2X3 antagonist 34    
P2X3 Receptor
    99.71%
JNJ-54175446        
P2X7 Receptor
99.30%
BX430      
P2X4 Receptor
  99.83%
Opiranserin hydrochloride    
P2X3 Receptor
    99.44%
Bullatine A        
P2X7 Receptor
≥98.0%
Eliapixant    
P2X3 Receptor
    99.95%
A-317491 sodium salt hydrate    
P2X3 Receptor
    99.88%
Lu AF27139        
P2X7 Receptor
99.71%
Gardenoside    
P2X3 Receptor
 
P2X7 Receptor
99.55%
Oxidized ATP trisodium salt        
P2X7 Receptor
≥98.0%
GW791343 dihydrochloride        
P2X7 Receptor, pIC50: 6.9-7.2
98.03%
EVT-401        
P2X7 Receptor
99.89%
Gefapixant citrate    
P2X3 Receptor
    99.23%
Opiranserin    
P2X3 Receptor
   
P2X4 antagonist-1      
P2X4 Receptor, IC50: 15 nM
  99.89%
P2X4 antagonist-2      
P2X4 Receptor, IC50: 24 nM
 
P2X7 receptor antagonist-3        
hP2X7R, IC50: 4.2 nM
rP2X7R, IC50: 6.8 nM
α,β-Methylene-ATP dilithium
p2x1 Receptor
 
P2X3 Receptor
 
P2X7 Receptor
PPADS
p2x1 Receptor, IC50: 68 nM
P2X2 Receptor, IC50: 214 nM
     
(S)-JNJ-54166060        
P2X7 Receptor
Minodronic acid-d4  
P2X2 Receptor
P2X3 Receptor
   
Blue FPG-A trisodium
p2x1 Receptor, IC50: 35.5 μM
       
P2X3 antagonist 38    
P2X3 Receptor, IC50: 0.132 μM
   
NF449
p2x1 Receptor
       
GW791343 trihydrochloride        
P2X7 Receptor, pIC50: 6.9-7.2