2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor Dopamine Receptor
  4. Quetiapine-d8 hemifumarate

Quetiapine-d8 hemifumarate  (Synonyms: 富马酸喹硫平 d8 (hemifumarate))

目录号: HY-B0031S3
产品使用指南

摩尔计算器

Quetiapine-d8 (hemifumarate) 是 Quetiapine hemifumarate 的氘代物。Quetiapine hemifumarate 是一种 5-HT 受体激动剂，对人 5-HT1A 的 pEC50 值为 4.77。Quetiapine hemifumarate 是多巴胺受体 (dopamine receptor) 拮抗剂，对人 D2 的 pIC50 值为 6.33。Quetiapine hemifumarate 对人 D2，HT1A，5-HT2A，5-HT2C 受体具有中高等亲和力，pKi 值为 7.25，5.74，7.54，5.55。具有抗抑郁和抗焦虑作用。

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Quetiapine-d<sub>8</sub> hemifumarate Chemical Structure

Quetiapine-d8 hemifumarate Chemical Structure

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Other Forms of Quetiapine-d8 hemifumarate:

Quetiapine-d8 hemifumarate 相关抗体

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Quetiapine-d8 (hemifumarate) is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor. Quetiapine hemifumarate has moderate to high affinity for the human D2, HT1A, 5-HT2A, 5-HT2C receptor with pKis of 7.25, 5.74, 7.54, 5.55. Antidepressant and anxiolytic effects[1].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Quetiapine-d8 hemifumarate 相关抗体:
分子量

507.63

Formula

C25H21D8N3O6S
非标记 CAS

111974-72-2
中文名称

富马酸喹硫平 d8 (hemifumarate)
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Quetiapine-d8 hemifumarate 相关分类

  • 摩尔计算器

  • 稀释计算器

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Quetiapine-d8 hemifumarate富马酸喹硫平 d8 (hemifumarate)5-HT ReceptorDopamine ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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