1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Dopamine Receptor
  4. Dopamine Receptor Inhibitors

Dopamine Receptor Inhibitors

Dopamine Receptor

D1 Receptor

D2 Receptor

D3 Receptor

D4 Receptor

D5 Receptor

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Dopamine Receptor Inhibitors, Agonists, Antagonists & Modulators
Product Name Dopamine Receptor D1 Receptor D2 Receptor D3 Receptor D4 Receptor D5 Receptor Purity
SCH-23390 hydrochloride  
D1 Receptor, Ki: 0.2 nM
     
D5 Receptor, Ki: 0.3 nM
99.91%
Haloperidol    
D2 Receptor
      99.73%
Clozapine    
D2 Receptor, Ki: 75 nM (Antagonist)
      99.97%
Olanzapine
Dopamine Receptor
          99.83%
Risperidone    
D2 Receptor, Ki: 5.9 nM
      99.92%
SKF 38393 hydrochloride  
D1 Receptor
        99.49%
Aripiprazole    
D2 Receptor
D3 Receptor
D4 Receptor
  99.95%
Cabergoline    
D2 Receptor
D3 Receptor
    99.86%
Bromocriptine mesylate    
D2 Receptor
      99.98%
WAY-100635        
D4 Receptor
  99.44%
Brexpiprazole    
D2L Receptor, Ki: 0.3 nM
      99.85%
Raclopride  
D1 Receptor, Ki: 18000 nM
D2 Receptor, Ki: 1.8 nM
D3 Receptor, Ki: 3.5 nM
D4 Receptor, Ki: 2400 nM
  99.83%
Sulpiride    
D2 Receptor
D3 Receptor
    99.75%
Penfluridol    
D2 Receptor
      99.93%
N-Methyldopamine hydrochloride  
D1 Receptor
        99.03%
Flunarizine dihydrochloride    
D2 Receptor
      99.87%
Domperidone    
D2 Receptor
      99.87%
WAY-100635 maleate        
D4 Receptor
  99.89%
Perphenazine    
D2 Receptor, Ki: 0.56 nM
D3 Receptor, Ki: 0.43 nM
D4 Receptor, Ki: 28.5 nM
  99.95%
Lurasidone    
D2 Receptor, IC50: 1.68 nM
      99.49%
Benztropine mesylate    
Human D2 Receptor
      99.92%
Cariprazine    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    99.83%
Paliperidone    
D2 Receptor
      99.69%
Ritanserin    
D2 Receptor, IC50: 70 nM
      99.68%
Nuciferine    
D2 Receptor, EC50: 64 nM
 
D4 Receptor, EC50: 2 μM
D5 Receptor, EC50: 2.6 μM
99.46%
Cariprazine hydrochloride    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    99.90%
Pramipexole    
D2 Receptor, Ki: 3.9 nM
D3 Receptor, Ki: 0.5 nM
D4 Receptor, Ki: 1.3 nM
  99.95%
Ziprasidone    
Rat D2 Receptor, Ki: 4.8 nM
      99.81%
Dihydrexidine hydrochloride  
D1 Receptor, IC50: 10 nM
        99.21%
Ropinirole hydrochloride    
D2 Receptor, Ki: 29 nM
hD2 Receptor, pEC50: 7.4
hD3 Receptor, pEC50: 8.4
hD4.4 Receptor, pEC50: 6.8
  99.85%
Rotigotine  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 4-15 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 4-15 nM
D5 Receptor, Ki: 4-15 nM
99.99%
SKF-82958 hydrobromide  
D1 Receptor
        99.82%
Loxapine  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
  99.69%
SKF 81297  
D1 Receptor
        99.86%
Piribedil    
D2 Receptor
D3 Receptor
    99.33%
A68930 hydrochloride  
D1 Receptor
        ≥98.0%
Loxapine succinate  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
  99.81%
Sumanirole maleate    
D2 Receptor
      99.78%
Flupentixol dihydrochloride  
D1 Receptor
D2 Receptor
      99.73%
Pramipexole dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
  99.73%
SKF 81297 hydrobromide  
D1 Receptor
        99.62%
Pergolide mesylate  
D1 Receptor
D2 Receptor
      99.92%
Rotigotine Hydrochloride  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 4-15 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 4-15 nM
D5 Receptor, Ki: 4-15 nM
99.65%
SKF-83566  
D1 Receptor
     
D5 Receptor
99.86%
Rotundine  
D1 Receptor, IC50: 166 nM
D2 Receptor, IC50: 1400 nM
D3 Receptor, IC50: 3300 nM
    99.96%
Flunarizine    
D2 Receptor
      99.93%
UNC9994 hydrochloride  
D1 Receptor, Ki: 4000 nM
D2 Receptor, Ki: 79 nM
D3 Receptor, Ki: 17 nM
D4 Receptor, Ki: 138 nM
  98.83%
Blonanserin  
D1 Receptor, Ki: 1070 nM
D2 Receptor, Ki: 0.142 nM
D3 Receptor, Ki: 0.494 nM
D4 Receptor, Ki: 150 nM
  99.62%
LY3154207  
D1 Receptor
        99.87%
Metoclopramide    
D2 Receptor, IC50: 483 nM
      99.94%
SB-277011 hydrochloride      
D3 Receptor, Ki: 10.7-11.2 nM
    98.54%
Ansofaxine hydrochloride
Dopamine Receptor, IC50: 491 nM
          99.72%
Chlorprothixene  
Human D1 Receptor, Ki: 18 nM
Human D2 Receptor, Ki: 2.96 nM
Human D3 Receptor, Ki: 4.56 nM
 
Human D5 Receptor, Ki: 9 nM
99.61%
Lurasidone Hydrochloride    
D2 Receptor, IC50: 1.68 nM
      99.96%
Buspirone    
Dopamine D2 receptor
      99.86%
Paliperidone palmitate    
D2 Receptor
      98.41%
Asenapine  
D1 Receptor, pKi: 8.9
D2 Receptor, pKi: 8.9
D3 Receptor, pKi: 9.4
D4 Receptor, pKi: 9.0
  99.62%
Ziprasidone hydrochloride monohydrate    
Rat D2 Receptor, Ki: 4.8 nM
      99.74%
Chlorprothixene hydrochloride  
Human D1 Receptor, Ki: 18 nM
Human D2 Receptor, Ki: 2.96 nM
Human D3 Receptor, Ki: 4.56 nM
 
Human D5 Receptor, Ki: 9 nM
99.91%
Sarizotan    
rD2 Receptor, IC50: 15.1 nM (rat)
hD2 Receptor, IC50: 17 nM
D3 Receptor, IC50: 6.8 nM (human)
hD4.2 Receptor, IC50: 2.4 nM
  98.74%
Pridopidine    
D2 Receptor
      99.85%
Talipexole dihydrochloride    
D2 Receptor
      99.80%
Thiethylperazine    
D2 Receptor
      99.41%
Ecopipam hydrochloride  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
99.46%
Tiapride hydrochloride    
D2 Receptor, IC50: 110-320 nM
D3 Receptor, IC50: 180 nM
    99.95%
Eticlopride hydrochloride    
D2 Receptor, Ki: 0.09 nM
      99.45%
Fluphenazine decanoate    
D2 Receptor
      ≥98.0%
Halopemide  
D1 Receptor
D2 Receptor
      99.65%
Pramipexole dihydrochloride hydrate    
D2 Receptor, Ki: 3.9 nM
D3 Receptor, Ki: 0.5 nM
D4 Receptor, Ki: 1.3 nM
  ≥98.0%
PD-168077 maleate        
D4 Receptor
  99.60%
L-745870    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 nM
Human D4 Receptor, Ki: 4.3 nM
  99.92%
Itopride hydrochloride    
D2 Receptor
      99.85%
Brilaroxazine    
D2 Receptor
D3 Receptor
D4 Receptor
  98.29%
SKF 83959  
D1 Receptor, Ki: 1.18 nM
D2 Receptor, Ki: 920 nM
D3 Receptor, Ki: 399 nM
 
D5 Receptor, Ki: 7.56 nM
98.94%
UNC9995    
D2 Receptor
      99.38%
Pericyazine    
D2 Receptor
      99.96%
(Rac)-Tavapadon  
D1 Receptor
        99.87%
Ocaperidone    
D2 Receptor, Ki: 0.75 nM
      99.93%
Bromperidol    
D2 Receptor
      98.48%
Iloperidone  
Rat D1 Receptor, Ki: 546 nM
Human D1 Receptor, Ki: 216 nM
Rat D2 Receptor, Ki: 54 nM
Human D3 Receptor, Ki: 7.1 nM
Human D4 Receptor, Ki: 25 nM
Human D5 Receptor, Ki: 319 nM
99.97%
Desmethyl cariprazine    
D2 Receptor, Ki: 0.49 nM
D3 Receptor, Ki: 0.085 nM
    98.06%
SKF 83822  
Rat D1 Receptor
        98.66%
A-77636 hydrochloride    
D2 Receptor
      ≥98.0%
Promazine hydrochloride    
D2 Receptor
      99.87%
ML417      
D3 Receptor, EC50: 38 nM
    99.50%
L-DOPA-2,5,6-d3      
D3 Receptor
    99.95%
Xaliproden hydrochloride    
D2 Receptor, IC50: 0.1-1 μM
      98.57%
Acetophenazine dimaleate    
D2 Receptor
      99.90%
Thiethylperazine dimaleate    
D2 Receptor
      99.72%
Brexpiprazole S-oxide-d8    
D2 Receptor, Ki: 0.3 nM
      98.72%
Didesmethyl cariprazine    
D2 Receptor
D3 Receptor
    99.79%
SKF 83959 hydrobromide  
D1 Receptor, Ki: 1.18 nM
D2 Receptor, Ki: 920 nM
D3 Receptor, Ki: 399 nM
 
D5 Receptor, Ki: 7.56 nM
99.86%
Metoclopramide hydrochloride hydrate    
D2 Receptor, IC50: 483 nM
      99.96%
PF-06256142  
Human D1 Receptor, EC50: 33 nM
        99.90%
Neuromedin N    
D2 Receptor
      99.61%
Naxagolide    
D2 Receptor
      99.81%
Quinelorane dihydrochloride    
D2 Receptor
D3 Receptor
    ≥99.0%
Spiramide  
D1 Receptor, Ki: 2530 nM
D2 Receptor, Ki: 3 nM
      99.23%
Propionylpromazine hydrochloride    
D2 Receptor
     
NGB 2904      
D3 Receptor, Ki: 1.4 nM
    98.28%
Perospirone hydrochloride  
D1 Receptor, Ki: 41 nM
D2 Receptor, Ki: 1.4 nM
      99.94%
Olanzapine-d3      
D3 Receptor
    99.09%
L-745870 hydrochloride    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 mM
Human D4 Receptor, Ki: 4.3 nM
  99.91%
Lumateperone  
D1 Receptor
D2 Receptor
      99.83%
Ecopipam hydrobromide  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
≥99.0%
Risperidone-d4    
D2 Receptor
      99.40%
GSK163090    
D2 Receptor, pKi: 6.3
D3 Receptor, pKi: 6.7
    99.77%
Cariprazine-d8      
D3 Receptor
    99.51%
Adoprazine    
D2 Receptor, pA2: 9.3
D2 Receptor, pKi: 8.4
D3 Receptor, pA2: 8.9
D3 Receptor, pKi: 8.4
D4 Receptor, pKi: 8.0
  98.60%
Carmoxirole hydrochloride    
D2 Receptor
      99.82%
(Rac)-PF-06256142  
Human D1 Receptor, EC50: 107 nM
        99.59%
Nemonapride    
D2 Receptor, Ki: 0.06 nM
      99.90%
ABT-724 trihydrochloride        
D4 Receptor
  99.05%
UNC9994    
D2 Receptor, Ki: 79 nM
D3 Receptor, Ki: 17 nM
D4 Receptor, Ki: 138 nM
  98.06%
(Rac)-Levomepromazine-d3 hydrochloride      
D3 Receptor
   
LE 300  
Human D1 Receptor, Ki: 1.9 nM
     
Human D5 Receptor, Ki: 7.5 nM
98.5%
Dopamine D4 receptor antagonist-1        
hD4.2 Receptor, Ki: 9.0 nM
  99.17%
Zuclopenthixol dihydrochloride    
D2 Receptor
      99.98%
Haloperidol-d4    
D2 Receptor
     
Spiperone hydrochloride  
D1 Receptor, Ki: ~350 nM
D2 Receptor, Ki: 0.06 nM
D3 Receptor, Ki: 0.6 nM
D4 Receptor, Ki: 0.08 nM
D5 Receptor, Ki: ~3500 nM
99.10%
PAOPA    
D2 Receptor
     
Lisuride    
D2 Receptor
      99.29%
S-14506 hydrochloride    
D2 Receptor
      99.92%
Fananserin        
D4 Receptor, Ki: 2.93 nM
  99.97%
(S)-Amisulpride    
D2 Receptor
D3 Receptor
    99.75%
SKF-83566 hydrobromide  
D1 Receptor
     
D5 Receptor
(-)-GSK598809 hydrochloride      
D3 Receptor
    99.64%
cis-(Z)-Flupentixol dihydrochloride    
D2 Receptor, Ki: 0.38 nM
     
SKF-75670 hydrobromide  
D1 Receptor
        99.83%
Brexpiprazole S-oxide    
D2 Receptor, Ki: 0.3 nM
     
SB-277011 dihydrochloride      
D3 Receptor
   
CY 208-243  
D1 Receptor
        99.98%
ST-836 hydrochloride    
D2 Receptor, Ki: 132 nM
D3 Receptor, Ki: 4.5 nM
    98.11%
Risperidone hydrochloride    
D2 Receptor, Ki: 5.9 nM
     
(Rac)-Rotigotine hydrochloride  
D1 Receptor, Ki: 83 nM
D2 Receptor, Ki: 13.5 nM
D3 Receptor, Ki: 0.71 nM
D4 Receptor, Ki: 3.9-15 nM
D5 Receptor, Ki: 5.4 nM
98.66%
Pardoprunox hydrochloride    
D2 Receptor, pEC50: 8
D3 Receptor, pEC50: 9.2
    99.46%
Ziprasidone hydrochloride    
Rat D2 Receptor, Ki: 4.8 nM
     
5-HT6/7 antagonist 1    
D2 Receptor
     
Clocapramine    
D2 Receptor
     
Propionylpromazine-d6 hydrochloride    
D2 Receptor
      99.78%
Blonanserin dihydrochloride  
D1 Receptor, Ki: 1070 nM
D2 Receptor, Ki: 0.142 nM
D3 Receptor, Ki: 0.494 nM
D4 Receptor, Ki: 150 nM
 
Mesdopetam      
D3 Receptor
   
Metoclopramide hydrochloride    
D2 Receptor, IC50: 483 nM
     
Thioridazine-d3 hydrochloride      
D3 Receptor
    99.19%
Amisulpride-d5 N-Oxide      
D3 Receptor
   
Iloperidone-d3      
D3 Receptor
   
Cabergoline-d5    
D2 Receptor
D3 Receptor
   
Amisulpride-d5      
D3 Receptor
    98.83%
Paliperidone-d4    
D2 Receptor
     
Pergolide-d7 mesylate    
D2 Receptor
     
Dopamine D3 receptor antagonist-2      
D3 Receptor, Ki: 2.16 nM
   
D4R antagonist-1        
D4 Receptor, IC50: 6.87 μM
 
Mesulergine hydrochloride
Dopamine Receptor
         
D5R agonist 1          
D5 Receptor, EC50: 269.7 nM
Bromocriptine-13C,d3    
D2 Receptor
D3 Receptor
   
Razpipadon  
D1 Receptor
       
Haloperidol-13C6    
D2 Receptor
     
D4R antagonist-2        
D4 Receptor
 
Blonanserin-d8    
D2 Receptor
     
Dopamine D4 receptor ligand 2    
D2 Receptor, IC50: >1000 nM
 
D4 Receptor, IC50: 0.057 nM
 
Agroclavine  
D1 Receptor
       
PD 119819
Dopamine Receptor
         
Carmoxirole    
D2 Receptor
     
Dopamine D2 receptor agonist-3    
D2 Receptor, EC50: 5 nM
D3 Receptor, EC50: >3.2 μM
   
SV 156    
Human D2 Receptor, Ki: 2.5 ± 0.4 nM
Human D3 Receptor, Ki: 96.9 ± 4.3 nM
Human D4 Receptor, Ki: 700 ± 56 nM
 
A-77636  
Dopamine D1 receptor, EC50: 1.1 nM
Dopamine D1 receptor, Ki: 39.8 nM
       
FAUC 346      
D3 Receptor, EC50: 1.5 nM
    99.90%
Tau-aggregation-IN-1    
D2 Receptor
D3 Receptor
   
BMY 28674    
D2 Receptor, IC50: 3.1 μM
D3 Receptor, IC50: 4.9 μM
D4 Receptor, IC50: 0.85 μM
 
SK609 hydrochloride      
Dopamine D3 receptor, EC50: 1109 nM
    99.83%
Fluphenazine decanoate dihydrochloride    
D2 Receptor
     
Ropinirole    
D2 Receptor, Ki: 29 nM
hD2 Receptor, pEC50: 7.4
hD3 Receptor, pEC50: 8.4
hD4.4 Receptor, pEC50: 6.8
 
Dopamine D3 receptor antagonist-1      
D3 Receptor
   
Dopamine D3 receptor ligand-1    
D2 Receptor, Ki: 715 nM
D3 Receptor, Ki: 8 nM
   
OS-3-106      
D3 Receptor, Ki: 0.2 nM
   
D3R ligand 1      
D3 Receptor, Ki: 66 nM
   
NGB 2904 hydrochloride      
D3 Receptor, Ki: 1.4
   
Brexpiprazole hydrochloride    
D2L Receptor, Ki: 0.3 nM
     
MOR agonist-2      
D3 Receptor
   
SUN-1334H free base      
Dopamine D3 receptor, IC50: 3.43 μM
   
Acetophenazine    
D2 Receptor
     
Benztropine    
D2 Receptor
     
Perphenazine dihydrochloride    
D2 Receptor, Ki: 0.56 nM
D3 Receptor, Ki: 0.43 nM
D4 Receptor, Ki: 28.5 nM
 
Promazine    
D2 Receptor
     
Asenapine citrate  
D1 Receptor, pKi: 8.9
D2 Receptor, pKi: 8.9
D3 Receptor, pKi: 9.4
D4 Receptor, pKi: 9.0
 
PD 158771    
hD2 Receptor, Ki: 42 nM
Human D3 Receptor, Ki: 13.7 nM
   
Cabergoline-d6    
D2 Receptor
D3 Receptor
   
BGC20-761    
Human D2 Receptor, Ki: 140 nM
     
Alizapride-13C,d3 hydrochloride      
D3 Receptor
   
Risperidone-d6    
D2 Receptor, Ki: 5.9 nM
     
SKF 38393 hydrobromide  
D1 Receptor, IC50: 110 nM
       
D4R antagonis-2        
D4 Receptor, IC50: 6.87 μM
 
A68930  
D1 Receptor
       
Dopamine D3 receptor ligand-3    
D2 Receptor, Ki: 353 nM
D3 Receptor, Ki: 3.6 nM
   
SCH-23390 maleate  
D1 Receptor, Ki: 0.2 nM
     
D5 Receptor, Ki: 0.3 nM
Itopride-d6 hydrochloride    
D2 Receptor
     
Piribedil dihydrochloride    
D2 Receptor
D3 Receptor
   
Cinitapride monotartrate    
D2 Receptor
     
Benztropine-13C,d3 mesylate    
D2 Receptor
D3 Receptor
   
PD 168568 dihydrochloride    
D2 Receptor, Ki: 1842 nM
D3 Receptor, Ki: 2682 nM
D4 Receptor, Ki: 8.8 nM
 
Ziprasidone mesylate    
Rat D2 Receptor, Ki: 4.8 nM
     
Dopamine D3 receptor ligand-4    
D2 Receptor, Ki: 7.43 nM
D3 Receptor, Ki: 0.5 nM
   
L-750667 triHydrochloride        
D4 Receptor, Ki: 0.51 nM
D4 Receptor, Kd: 0.16 nM
 
L-745870 trihydrochloride    
D2 Receptor, Ki: 960 nM
D3 Receptor, Ki: 2300 nM
Human D4 Receptor, Ki: 4.3 nM
 
(Rac)-Rotigotine-d7 hydrochloride  
D1 Receptor
 
D3 Receptor
D4 Receptor
 
Levosulpiride-d3      
D3 Receptor
    99.79%
Asenapine-13C,d3 hydrochloride      
D3 Receptor
D4 Receptor
 
(S)-Remoxipride  
D1 Receptor, IC50: >100 μM
D2 Receptor, IC50: 1.57 μM
     
PD 168568    
D2 Receptor, Ki: 1842 nM
D3 Receptor, Ki: 2682 nM
D4 Receptor, Ki: 8.8 nM
 
Blonanserin-d5    
D2 Receptor
     
Aripiprazole monohydrate    
D2 Receptor
D3 Receptor
D4 Receptor
 
DETQ  
Human D1 Receptor, EC50: 5.8 nM
       
Itopride    
D2 Receptor
     
Pramipexole-d7 dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
 
FGH31        
Dopamine D4 receptor, Ki: 1.6 nM
 
Ziprasidone mesylate trihydrate    
Rat D2 Receptor, Ki: 4.8 nM
     
Ordopidine    
D2 Receptor
     
Asimilobine
Dopamine Receptor
         
Piribedil hydrochloride    
D2 Receptor
D3 Receptor
   
NEO 376
Dopamine Receptor
          99.23%
Loxapine hydrochloride  
Human D1 Receptor
Human D2 Receptor
 
Human D4 Receptor
 
PNU-177864 hydrochloride      
D3 Receptor
   
Bromperidol hydrochloride    
D2 Receptor
      99.96%
Bifeprunox    
D2 Receptor, pKi: 8.83 (striatum)
     
Antipsychotic agent-2    
D2 Receptor, Kb: 45.7 nM
     
BP 897    
D2 Receptor
D3 Receptor
   
A-69024  
D1 Receptor, Ki: 12.6 nM
D2 Receptor, Ki: 1290 nM
     
Cyclo(glycyl-L-leucyl)
Dopamine Receptor
         
Dopamine D3 receptor ligand-2    
D2 Receptor, Ki: 1228 nM
D3 Receptor, Ki: 11.4 nM
   
SKF83822 hydrobromide  
D1 Receptor
       
Haloperidol-d4-1    
D2 Receptor
      ≥98.0%
Pramipexole-d5 dihydrochloride    
D2 Receptor
D3 Receptor
D4 Receptor
 
Flupentixol  
D1 Receptor
D2 Receptor
     
SB-414796    
D2 Receptor, Ki: 400 nM
D3 Receptor, Ki: 4 nM
   
Tiapride    
D2 Receptor, IC50: 110-320 nM
D3 Receptor, IC50: 180 nM
   
FAUC 213    
hD2 Receptor, Ki: 3.4 μM
hD3 Receptor, Ki: 5.3 μM
hD4.4 Receptor, Ki: 2.2 nM
  99.86%
PNU-96415E        
D4 Receptor
 
Ecopipam  
D1 Receptor, Ki: 1.2 nM
D2 Receptor, Ki: 980 nM
 
D4 Receptor, Ki: 5520 nM
D5 Receptor, Ki: 2.0 nM
Raclopride tartrate  
D1 Receptor, Ki: 18000 nM
D2 Receptor, Ki: 1.8 nM
D3 Receptor, Ki: 3.5 nM
D4 Receptor, Ki: 2400 nM
 
Sonepiprazole    
rD2 Receptor, Ki: 5147 nM
 
rD4 Receptor, Ki: 3.6 nM
  99.84%
PG01037 dihydrochloride      
D3 Receptor, Ki: 0.7 nM
   
BL-1020 mesylate    
D2L Receptor, Ki: 0.066 nM
     
FR 64822    
D2 Receptor
     
Haloperidol-d4 N-Oxide    
D2 Receptor
     
Risperidone mesylate    
D2 Receptor, Ki: 5.9 nM
     
U-101958 maleate    
D2 Receptor, IC50: 1980 nM
D3 Receptor, IC50: 552 nM
D4 Receptor, IC50: 2.7 nM
 
PD 118717    
D2 Receptor
     
ADX-10061  
D1 Receptor, Ki: 5.8 nM
D2 Receptor, Ki: > >10 000 nM
     
BRD5814    
D2 Receptor
     
Iloperidone hydrochloride  
Rat D1 Receptor, Ki: 546 nM
Human D1 Receptor, Ki: 216 nM
Rat D2 Receptor, Ki: 54 nM
Human D3 Receptor, Ki: 7.1 nM
Human D4 Receptor, Ki: 25 nM
Human D5 Receptor, Ki: 319 nM
FAUC-312  
Dopamine D1 receptor, Ki: 29000 nM
Dopamine D2 receptor, Ki: 25000 nM
Dopamine D3 receptor, Ki: 13000 nM
Dopamine D4 receptor, Ki: 1.5 nM
 
Aplindore    
D2 Receptor, pKi: 9.1
     
Sumanirole    
D2 Receptor
     
Pardoprunox    
D2 Receptor, pEC50: 8
D3 Receptor, pEC50: 9.2
   
7-Hydroxy-PIPAT      
D3 Receptor, Ki: 0.99 nM
   
Sarizotan dihydrochloride      
Human D3 Receptor, IC50: 6.8 nM
   
Pimozide-d5 N-Oxide  
D1 Receptor
 
D3 Receptor
   
Abaperidone    
D2 Receptor, IC50: 17 nM
     
NRA-0160      
D3 Receptor, Ki: 39 nM
D4 Receptor, Ki: 0.48 nM
 
SKF 83509    
D2 Receptor, Ki: 70.2 nM
     
Dexpramipexole-d3 dihydrochloride      
D3 Receptor
   
Clozapine hydrochloride    
D2 Receptor, Ki: 75 nM
     
Raclopride-d5 hydrochloride      
D3 Receptor
    99.82%
Clocapramine dihydrochloride hydrate    
D2 Receptor
     
(-)-GSK598809      
D3 Receptor
   
BP 897 hydrochloride    
D2 Receptor
D3 Receptor
    99.84%