2. Membrane Transporter/Ion Channel
  3. Sodium Channel Potassium Channel
  4. Eleclazine

Eleclazine  (Synonyms: GS-6615)

目录号: HY-16738
产品使用指南

摩尔计算器

Eleclazine (GS 6615) 是一种具有选择性的心脏晚期钠电流 (sodium current) 抑制剂和钾电流 (potassium current) 的弱抑制剂，IC50 值分别为 <1 μM 和约 14.2 μM。在猪模型中，Eleclazine 对自发性心房早搏、复极交替和异质性以及心房纤颤同时具有保护作用。Eleclazine 可用于心律失常的研究。

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Eleclazine Chemical Structure

Eleclazine Chemical Structure

CAS No. : 1443211-72-0

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Eleclazine 的其他形式现货产品:

Other Forms of Eleclazine:

Eleclazine 相关抗体

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Eleclazine (GS 6615) is a selective cardiac late sodium current inhibitor and a weak inhibitor of potassium current with IC50 of <1 μM and approximately 14.2 μM, respectively. Eleclazine shows concurrent protection against autonomically induced atrial premature beats, repolarization alternans and heterogeneity, and atrial fibrillation in porcine model. Eleclazine can be used to research cardiac arrhythmias[1][2][3].

分子量

415.37

Formula

C21H16F3N3O3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Eleclazine 相关分类

  • 摩尔计算器

  • 稀释计算器

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Eleclazine1443211-72-0GS-6615GS6615GS 6615Sodium ChannelPotassium ChannelNa channelsNa+ channelsKcsAInhibitorinhibitorinhibit

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