2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. Mu opioid receptor antagonist 2

Mu opioid receptor antagonist 2 

目录号: HY-144607
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摩尔计算器

Mu opioid receptor antagonist 2 (compound 25) 是一种有效且具有选择性和血脑屏障渗透性的 μ 阿片受体 (MOR) 拮抗剂，Ki 为 0.37 nM，EC50 为 0.44 nM。Mu opioid receptor antagonist 2 对吗啡具有显著的中枢神经系统拮抗作用，与 Naloxone 相比，其诱发戒断症状较少。Mu opioid receptor antagonist 2 可用于阿片类活性分子使用障碍 (OUD) 的研究。

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Mu opioid receptor antagonist 2 Chemical Structure

Mu opioid receptor antagonist 2 Chemical Structure

CAS No. : 2773925-64-5

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Mu opioid receptor antagonist 2 相关抗体

Top Publications Citing Use of Products

查看 Opioid Receptor 亚型特异性产品:

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μ Opioid Receptor/MOR κ Opioid Receptor/KOR δ Opioid Receptor/DOR NOP Receptor/ORL1

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  • 参考文献

生物活性

Mu opioid receptor antagonist 2 (compound 25) is a potent, selective and blood-brain barrier (BBB) penetrant μ opioid receptor (MOR) antagonist with a Ki of 0.37 nM and an EC50 of 0.44 nM. Mu opioid receptor antagonist 2 has remarkable CNS antagonism against morphine, and precipitated fewer withdrawal symptoms than Naloxone. Mu opioid receptor antagonist 2 can be used for researching opioid use disorders (OUD)[1].

IC50 & Target

μ Opioid Receptor/MOR

 

分子量

452.57

Formula

C25H28N2O4S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Mu opioid receptor antagonist 2 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Mu opioid receptor antagonist 22773925-64-5Mu opioid receptor antagonist2Mu opioid receptor antagonist-2Opioid Receptorμ opioid receptorOpioid use disordersBlood-brain barrier penetrantWithdrawal symptomsInhibitorinhibitorinhibit

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