COS-1
|
EC50 |
> 1000 nM
Compound: 1, GW-501516
|
Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene assay
Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene assay
|
[PMID: 22051054]
|
COS-1
|
EC50 |
0.5 nM
Compound: 1, GW501516
|
Agonist activity at pSG5-Gal4-tagged human PPAR-beta/delta ligand binding domain expressed in COS1 cells assessed as receptor activation incubated for 19 hrs by pGL3-5XUAS-SV40 luciferase reporter gene assay
Agonist activity at pSG5-Gal4-tagged human PPAR-beta/delta ligand binding domain expressed in COS1 cells assessed as receptor activation incubated for 19 hrs by pGL3-5XUAS-SV40 luciferase reporter gene assay
|
[PMID: 25768705]
|
COS-1
|
EC50 |
2.9 nM
Compound: 1, GW-501516
|
Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analysis
Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analysis
|
[PMID: 22051054]
|
COS-1
|
EC50 |
912 nM
Compound: 1, GW-501516
|
Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analysis
Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometric analysis
|
[PMID: 22051054]
|
COS-7
|
EC50 |
|
Activity at PPARbeta/delta by luciferase reporter gene transactivation assay in COS7 cells
Activity at PPARbeta/delta by luciferase reporter gene transactivation assay in COS7 cells
|
[PMID: 16797985]
|
COS-7
|
EC50 |
10000 nM
Compound: GW-501516
|
Activity at PPARalpha by luciferase reporter gene transactivation assay in COS7 cells
Activity at PPARalpha by luciferase reporter gene transactivation assay in COS7 cells
|
[PMID: 16797985]
|
COS-7
|
EC50 |
10000 nM
Compound: GW-501516
|
Activity at PPARgamma by luciferase reporter gene transactivation assay in COS7 cells
Activity at PPARgamma by luciferase reporter gene transactivation assay in COS7 cells
|
[PMID: 16797985]
|
CV-1
|
EC50 |
> 1.2 μM
Compound: GW501516
|
Transactivation activity at human PPARgamma expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
Transactivation activity at human PPARgamma expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
|
[PMID: 22534184]
|
CV-1
|
EC50 |
0.001 μM
Compound: 1, GW-501516
|
Agonist potency at PPARdelta in CV1 cells by cell based transient transfection assay
Agonist potency at PPARdelta in CV1 cells by cell based transient transfection assay
|
[PMID: 17243659]
|
CV-1
|
EC50 |
0.0012 μM
Compound: GW501516
|
Transactivation of human PPARdelta expressed in african green monkey CV1 cells by luciferase reporter gene assay
Transactivation of human PPARdelta expressed in african green monkey CV1 cells by luciferase reporter gene assay
|
[PMID: 22579420]
|
CV-1
|
EC50 |
0.0017 μM
Compound: 1, GW-501516
|
Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
Agonist activity at human PPARdelta-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
|
[PMID: 21515063]
|
CV-1
|
EC50 |
0.0017 μM
Compound: GW-501516
|
Transactivation of Gal4-fused human PPARdelta DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
Transactivation of Gal4-fused human PPARdelta DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
|
[PMID: 21112784]
|
CV-1
|
EC50 |
0.99 μM
Compound: 1, GW-501516
|
Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
Agonist activity at human PPARalpha-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
|
[PMID: 21515063]
|
CV-1
|
EC50 |
0.99 μM
Compound: GW-501516
|
Transactivation of Gal4-fused human PPARalpha DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
Transactivation of Gal4-fused human PPARalpha DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
|
[PMID: 21112784]
|
CV-1
|
EC50 |
1.888 μM
Compound: 1, GW-501516
|
Agonist potency at PPARalpha in CV1 cells by cell based transient transfection assay
Agonist potency at PPARalpha in CV1 cells by cell based transient transfection assay
|
[PMID: 17243659]
|
CV-1
|
EC50 |
2.5 nM
Compound: GW501516
|
Transactivation activity at human PPARdelta expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
Transactivation activity at human PPARdelta expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
|
[PMID: 22534184]
|
CV-1
|
EC50 |
229 nM
Compound: GW501516
|
Transactivation activity at human PPARalpha expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
Transactivation activity at human PPARalpha expressed in african green monkey CV1 cells after 24 hrs by luciferase reporter gene assay
|
[PMID: 22534184]
|
CV-1
|
EC50 |
4.1 μM
Compound: 1, GW-501516
|
Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
Agonist activity at human PPARgamma-LBD expressed in CV1 cells co-transfected with Gal4 after 40 hrs by luciferase based transactivation assay
|
[PMID: 21515063]
|
CV-1
|
EC50 |
4.1 μM
Compound: GW-501516
|
Transactivation of Gal4-fused human PPARgamma DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
Transactivation of Gal4-fused human PPARgamma DNA binding domain expressed in african green monkey CV1 cells by luciferase reporter gene assay
|
[PMID: 21112784]
|
CV-1
|
EC50 |
8.9 μM
Compound: 1, GW-501516
|
Agonist potency at PPARgamma in CV1 cells by cell based transient transfection assay
Agonist potency at PPARgamma in CV1 cells by cell based transient transfection assay
|
[PMID: 17243659]
|
HEK293
|
EC50 |
> 10 μM
Compound: GW-501516
|
Activity at human adipose tissue PPAR gamma expressed in HEK293 cells by PPAR-GAL4 transactivation assay
Activity at human adipose tissue PPAR gamma expressed in HEK293 cells by PPAR-GAL4 transactivation assay
|
[PMID: 17343371]
|
HEK293
|
EC50 |
0.002 μM
Compound: 1, GW-501516
|
Agonist activity at Gal4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assay
Agonist activity at Gal4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assay
|
[PMID: 21094606]
|
HEK293
|
EC50 |
0.0044 μM
Compound: GW501516
|
Agonist activity at GAL4N fused human PPARdelta LBD expressed in HEK293 cells co-expressing TK-MH100x4-Luc after 24 hrs by luciferase reporter gene assay
Agonist activity at GAL4N fused human PPARdelta LBD expressed in HEK293 cells co-expressing TK-MH100x4-Luc after 24 hrs by luciferase reporter gene assay
|
[PMID: 28539218]
|
HEK293
|
EC50 |
0.0059 μM
Compound: GW501516
|
Agonist activity at N-terminal Gal4 fused human PPARdelta LBD transfected in HEK293 cells after 24 hrs by luciferase reporter gene assay
Agonist activity at N-terminal Gal4 fused human PPARdelta LBD transfected in HEK293 cells after 24 hrs by luciferase reporter gene assay
|
[PMID: 27622746]
|
HEK293
|
EC50 |
0.0059 μM
Compound: GW501516
|
Agonist activity at GAL4-tagged human PPARdelta ligand binding domain chimeric receptor expressed in HEK293 cells after 24 hrs by luciferase reporter gene assay
Agonist activity at GAL4-tagged human PPARdelta ligand binding domain chimeric receptor expressed in HEK293 cells after 24 hrs by luciferase reporter gene assay
|
[PMID: 27591006]
|
HEK293
|
EC50 |
0.0079 μM
Compound: GW-501516
|
Activity at human placenta PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assay
Activity at human placenta PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assay
|
[PMID: 17343371]
|
HEK293
|
EC50 |
0.054 μM
Compound: GW-501516
|
Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assay
Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assay
|
[PMID: 17343371]
|
HEK293
|
EC50 |
0.085 μM
Compound: GW-501516
|
Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assay
Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assay
|
[PMID: 17524643]
|
HEK293
|
EC50 |
0.18 nM
Compound: GW501516
|
Agonist activity at human PPARbeta expressed in HEK293 cells by luciferase reporter gene assay
Agonist activity at human PPARbeta expressed in HEK293 cells by luciferase reporter gene assay
|
[PMID: 25305688]
|
HEK293
|
EC50 |
3.9 μM
Compound: GW-501516
|
Activity at human liver PPAR alpha expressed in HEK293 cells by PPAR-GAL4 transactivation assay
Activity at human liver PPAR alpha expressed in HEK293 cells by PPAR-GAL4 transactivation assay
|
[PMID: 17343371]
|
HeLa
|
EC50 |
> 10000 nM
Compound: 27, GW-501516
|
Agonist activity at PPARalpha ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
Agonist activity at PPARalpha ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
|
[PMID: 19275963]
|
HeLa
|
EC50 |
> 10000 nM
Compound: 27, GW-501516
|
Agonist activity at PPARgamma ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
Agonist activity at PPARgamma ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
|
[PMID: 19275963]
|
HeLa
|
EC50 |
8 nM
Compound: 27, GW-501516
|
Agonist activity at PPARdelta ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
Agonist activity at PPARdelta ligand binding domain expressed in human HeLa cells co-transfected with Gal4-DBD assessed as transcriptional activation by Gal4 response element-driven luciferase reporter gene assay
|
[PMID: 19275963]
|
HepG2
|
EC50 |
0.0012 μM
Compound: GW-501516
|
Agonist activity at human PPARdelta expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
Agonist activity at human PPARdelta expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
|
[PMID: 21215640]
|
HepG2
|
EC50 |
0.8 μM
Compound: GW-501516
|
Agonist activity at human PPARgamma expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
Agonist activity at human PPARgamma expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
|
[PMID: 21215640]
|
HepG2
|
EC50 |
1.1 μM
Compound: GW-501516
|
Agonist activity at human PPARalpha expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
Agonist activity at human PPARalpha expressed in HepG2 cells co-transfected with PPRE3-TK-luc assessed as beta-galactosidase activity after 20 to 22 hrs by luciferase based transactivation assay
|
[PMID: 21215640]
|
HepG2
|
EC50 |
|
Agonist activity at human PPARdelta in HepG2 cells by GAL4-luciferase reporter gene assay
Agonist activity at human PPARdelta in HepG2 cells by GAL4-luciferase reporter gene assay
|
[PMID: 17512197]
|