2. Neuronal Signaling GPCR/G Protein
  3. Cholinesterase (ChE) 5-HT Receptor
  4. Flucopride

Flucopride (Compound 4a) 是一种 AChE 抑制剂 (IC50: 24 nM)，也是一种部分 5-HT4R 激动剂 (对 (h)5-HT4R 的 Ki4R 的 COS-7 细胞中 APP 的非淀粉样变性加工 (EC50: 23.0 nM)。Flucopride 可能具有良好的胃肠道 (GIT) 渗透性和血脑屏障 (BBB) 跨膜渗透性 (PAMPA 实验测定)。

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Flucopride Chemical Structure

Flucopride Chemical Structure

CAS No. : 1639925-34-0

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Flucopride 相关抗体

Top Publications Citing Use of Products

查看 Cholinesterase (ChE) 亚型特异性产品:

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AChE BChE

查看 5-HT Receptor 亚型特异性产品:

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5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Flucopride (Compound 4a) is an AChE inhibitor (IC50: 24 nM), and a partial 5-HT4R agonist (Ki4R (EC50: 23.0 nM). Flucopride may has good gastrointestinal track (GIT) penetration, and blood-brain barrier (BBB) cross-membrane penetration (PAMPA assay)[1].

IC50 & Target[1]

AChE

24 nM (IC50)

huamn 5-HT4(c) Receptor

9.6 nM (Ki)

分子量

376.51

Formula

C22H33FN2O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Flucopride 相关分类

  • 摩尔计算器

  • 稀释计算器

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Flucopride1639925-34-0Cholinesterase (ChE)5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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